Recent Advances and New Strategies in Targeting Plk1 for Anticancer Therapy
Lee, Kyung S, Burke, Terrence R, Park, Jung-Eun, Bang, Jeong K, Lee, Eunhye
Published in Trends in pharmacological sciences (Regular ed.) (01.12.2015)
Published in Trends in pharmacological sciences (Regular ed.) (01.12.2015)
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Journal Article
Examination of aminophenol-containing compounds designed as antiproliferative agents and potential atypical retinoids
Chingle, Ramesh M., Imai, Masahiko, Altman, Sarah, Saito, Daisuke, Takahashi, Noriko, Burke, Terrence R.
Published in Bioorganic & medicinal chemistry (15.03.2023)
Published in Bioorganic & medicinal chemistry (15.03.2023)
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Journal Article
Enhancing polo-like kinase 1 selectivity of polo-box domain-binding peptides
Zhao, Xue Zhi, Hymel, David, Burke, Terrence R.
Published in Bioorganic & medicinal chemistry (01.10.2017)
Published in Bioorganic & medicinal chemistry (01.10.2017)
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Journal Article
Effects on polo-like kinase 1 polo-box domain binding affinities of peptides incurred by structural variation at the phosphoamino acid position
Qian, Wenjian, Park, Jung-Eun, Liu, Fa, Lee, Kyung S., Burke, Terrence R.
Published in Bioorganic & medicinal chemistry (15.07.2013)
Published in Bioorganic & medicinal chemistry (15.07.2013)
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Journal Article
Non-proteinogenic amino acids in the pThr-2 position of a pentamer peptide that confer high binding affinity for the polo box domain (PBD) of polo-like kinase 1 (Plk1)
Qian, Wen-Jian, Park, Jung-Eun, Lee, Kyung S., Burke, Terrence R.
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
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Journal Article
6,7-Dihydroxy-1-oxoisoindoline-4-sulfonamide-containing HIV-1 integrase inhibitors
Zhao, Xue Zhi, Maddali, Kasthuraiah, Smith, Steven J., Métifiot, Mathieu, Johnson, Barry C., Marchand, Christophe, Hughes, Stephen H., Pommier, Yves, Burke, Terrence R.
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
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Journal Article
Development of tricyclic hydroxy-1H-pyrrolopyridine-trione containing HIV-1 integrase inhibitors
Zhao, Xue Zhi, Maddali, Kasthuraiah, Metifiot, Mathieu, Smith, Steven J, Christie Vu, B, Marchand, Christophe, Hughes, Stephen H, Pommier, Yves, Burke, Terrence R., Jr
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Journal Article
Examination of halogen substituent effects on HIV-1 integrase inhibitors derived from 2,3-dihydro-6,7-dihydroxy-1H-isoindol-1-ones and 4,5-dihydroxy-1H-isoindole-1,3(2H)-diones
XUE ZHI ZHAO, MADDALI, Kasthuraiah, VU, B. Christie, MARCHAND, Christophe, HUGHES, Stephen H, POMMIER, Yves, BURKE, Terrence R
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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Journal Article
Development of antiproliferative phenylmaleimides that activate the unfolded protein response
Muus, Ulrike, Hose, Curtis, Yao, Wei, Kosakowska-Cholody, Teresa, Farnsworth, David, Dyba, Marzena, Lountos, George T., Waugh, David S., Monks, Anne, Burke, Terrence R., Michejda, Christopher J.
Published in Bioorganic & medicinal chemistry (15.06.2010)
Published in Bioorganic & medicinal chemistry (15.06.2010)
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Journal Article
A rapid oxime linker-based library approach to identification of bivalent inhibitors of the Yersinia pestis protein-tyrosine phosphatase, YopH
Liu, Fa, Hakami, Ramin Mollaaghababa, Dyas, Beverly, Bahta, Medhanit, Lountos, George T., Waugh, David S., Ulrich, Robert G., Burke, Terrence R.
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
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Journal Article
Application of ring-closing metathesis macrocyclization to the development of Tsg101-binding antagonists
Liu, Fa, Stephen, Andrew G., Waheed, Abdul A., Freed, Eric O., Fisher, Robert J., Burke, Terrence R.
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
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Journal Article
Application of azide–alkyne cycloaddition ‘click chemistry’ for the synthesis of Grb2 SH2 domain-binding macrocycles
Choi, Won Jun, Shi, Zhen-Dan, Worthy, Karen M., Bindu, Lakshman, Karki, Rajeshri G., Nicklaus, Marc C., Fisher, Robert J., Burke, Terrence R.
Published in Bioorganic & medicinal chemistry letters (15.10.2006)
Published in Bioorganic & medicinal chemistry letters (15.10.2006)
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Journal Article
Crystal Structures of a High-affinity Macrocyclic Peptide Mimetic in Complex with the Grb2 SH2 Domain
Phan, Jason, Shi, Zhen-Dan, Burke, Terrence R., Waugh, David S.
Published in Journal of molecular biology (14.10.2005)
Published in Journal of molecular biology (14.10.2005)
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