Potent, Orally Active Heterocycle-Based Combretastatin A-4 Analogues: Synthesis, Structure−Activity Relationship, Pharmacokinetics, and In Vivo Antitumor Activity Evaluation
Wang, Le, Woods, Keith W, Li, Qun, Barr, Kenneth J, McCroskey, Richard W, Hannick, Steven M, Gherke, Laura, Credo, R. Bruce, Hui, Yu-Hua, Marsh, Kennan, Warner, Robert, Lee, Jang Y, Zielinski-Mozng, Nicolette, Frost, David, Rosenberg, Saul H, Sham, Hing L
Published in Journal of medicinal chemistry (11.04.2002)
Published in Journal of medicinal chemistry (11.04.2002)
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Syntheses of Potent, Selective, and Orally Bioavailable Indazole-Pyridine Series of Protein Kinase B/Akt Inhibitors with Reduced Hypotension
Zhu, Gui-Dong, Gandhi, Viraj B, Gong, Jianchun, Thomas, Sheela, Woods, Keith W, Song, Xiaohong, Li, Tongmei, Diebold, R. Bruce, Luo, Yan, Liu, Xuesong, Guan, Ran, Klinghofer, Vered, Johnson, Eric F, Bouska, Jennifer, Olson, Amanda, Marsh, Kennan C, Stoll, Vincent S, Mamo, Mulugeta, Polakowski, James, Campbell, Thomas J, Martin, Ruth L, Gintant, Gary A, Penning, Thomas D, Li, Qun, Rosenberg, Saul H, Giranda, Vincent L
Published in Journal of medicinal chemistry (28.06.2007)
Published in Journal of medicinal chemistry (28.06.2007)
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Heteroarylmethoxyphenylalkoxyiminoalkylcarboxylic Acids as Leukotriene Biosynthesis Inhibitors
Kolasa, Teodozyj, Gunn, David E, Bhatia, Pramila, Woods, Keith W, Gane, Todd, Stewart, Andrew O, Bouska, Jennifer B, Harris, Richard R, Hulkower, Keren I, Malo, Peter E, Bell, Randy L, Carter, George W, Brooks, Clint D. W
Published in Journal of medicinal chemistry (24.02.2000)
Published in Journal of medicinal chemistry (24.02.2000)
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Journal Article
Potent, Orally Active Heterocycle-Based Combretastatin A-4 Analogues: Synthesis, Structure−Activity Relationship, Pharmacokinetics, and In Vivo Antitumor Activity Evaluation
Wang, Le, Woods, Keith W, Li, Qun, Barr, Kenneth J, McCroskey, Richard W, Hannick, Steven M, Gherke, Laura, Credo, R. Bruce, Hui, Yu-Hua, Marsh, Kennan, Warner, Robert, Lee, Jang Y, Zielinski-Mozng, Nicolette, Frost, David, Rosenberg, Saul H, Sham, Hing L
Published in Journal of medicinal chemistry (24.10.2002)
Published in Journal of medicinal chemistry (24.10.2002)
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Journal Article
Studies directed toward the design of orally active renin inhibitors. 1. Some factors influencing the absorption of small peptides
Rosenberg, Saul H, Spina, Kenneth P, Woods, Keith W, Polakowski, Jim, Martin, Donald L, Yao, Zhengli, Stein, Herman H, Cohen, Jerome, Barlow, Jennifer L
Published in Journal of medicinal chemistry (19.02.1993)
Published in Journal of medicinal chemistry (19.02.1993)
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Water-soluble renin inhibitors: design of a subnanomolar inhibitor with a prolonged duration of action
Rosenberg, Saul H, Woods, Keith W, Sham, Hing L, Kleinert, Hollis D, Martin, Donald L, Stein, Herman, Cohen, Jerome, Egan, David A, Bopp, Barbara
Published in Journal of medicinal chemistry (01.07.1990)
Published in Journal of medicinal chemistry (01.07.1990)
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Journal Article
Potent, low molecular weight renin inhibitors containing a C-terminal heterocycle: hydrogen bonding at the active site
Rosenberg, Saul H, Dellaria, Joseph F, Kempf, Dale J, Hutchins, Charles W, Woods, Keith W, Maki, Robert G, De Lara, Ed, Spina, Kenneth P, Stein, Herman H
Published in Journal of medicinal chemistry (01.06.1990)
Published in Journal of medicinal chemistry (01.06.1990)
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Novel renin inhibitors containing analogs of statine retro-inverted at the C-termini. Specificity at the P2 histidine site
Rosenberg, Saul H, Plattner, Jacob J, Woods, Keith W, Stein, Herman H, Marcotte, Patrick A, Cohen, Jerome, Perun, Thomas J
Published in Journal of medicinal chemistry (01.07.1987)
Published in Journal of medicinal chemistry (01.07.1987)
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Journal Article
Azido glycols: potent, low molecular weight renin inhibitors containing an unusual post scissile site residue
Rosenberg, Saul H, Woods, Keith W, Kleinert, Hollis D, Stein, Herman, Nellans, Hugh N, Hoffman, Daniel J, Spanton, Stephen G, Pyter, Richard A, Cohen, Jerome
Published in Journal of medicinal chemistry (01.06.1989)
Published in Journal of medicinal chemistry (01.06.1989)
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