Clavulanic acid: A competitive inhibitor of beta-lactamases with novel anxiolytic-like activity and minimal side effects
Kim, Deog J., King, Jean A., Zuccarelli, Lisa, Ferris, Craig F., Koppel, Gary A., Snowdon, Charles T., Ahn, Chang H.
Published in Pharmacology, biochemistry and behavior (01.08.2009)
Published in Pharmacology, biochemistry and behavior (01.08.2009)
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Orally active vasopressin V1a receptor antagonist, SRX251, selectively blocks aggressive behavior
Ferris, Craig F., Lu, Shi-fang, Messenger, Tara, Guillon, Christophe D., Heindel, Ned, Miller, Marvin, Koppel, Gary, Robert Bruns, F., Simon, Neal G.
Published in Pharmacology, biochemistry and behavior (01.02.2006)
Published in Pharmacology, biochemistry and behavior (01.02.2006)
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Azetidinones as vasopressin V1a antagonists
Guillon, Christophe D., Koppel, Gary A., Brownstein, Michael J., Chaney, Michael O., Ferris, Craig F., Lu, Shi-fang, Fabio, Karine M., Miller, Marvin J., Heindel, Ned D., Hunden, David C., Cooper, Robin D.G., Kaldor, Stephen W., Skelton, Jeffrey J., Dressman, Bruce A., Clay, Michael P., Steinberg, Mitchell I., Bruns, Robert F., Simon, Neal G.
Published in Bioorganic & medicinal chemistry (01.03.2007)
Published in Bioorganic & medicinal chemistry (01.03.2007)
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Vasopressin antagonists as anxiolytics and antidepressants: recent developments
Simon, Neal G, Guillon, Christophe, Fabio, Karine, Heindel, Ned D, Lu, Shi-fang, Miller, Marvin, Ferris, Craig F, Brownstein, Michael J, Garripa, Carrie, Koppel, Gary A
Published in Recent patents on CNS drug discovery (01.06.2008)
Published in Recent patents on CNS drug discovery (01.06.2008)
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LY320135, a Novel Cannabinoid CB1 Receptor Antagonist, Unmasks Coupling of the CB1 Receptor to Stimulation of cAMP Accumulation
Felder, C C, Joyce, K E, Briley, E M, Glass, M, Mackie, K P, Fahey, K J, Cullinan, G J, Hunden, D C, Johnson, D W, Chaney, M O, Koppel, G A, Brownstein, M
Published in The Journal of pharmacology and experimental therapeutics (01.01.1998)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.1998)
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Isolation and measurement of the endogenous cannabinoid receptor agonist, anandamide, in brain and peripheral tissues of human and rat
Felder, Christian C., Nielsen, Amie, Briley, Eileen M., Palkovits, Miklós, Priller, Joseph, Axelrod, Julius, Nguyen, Duy N., Richardson, John M., Riggin, Ralph M., Koppel, Gary A., Paul, Steven M., Becker, Gerald W.
Published in FEBS letters (16.09.1996)
Published in FEBS letters (16.09.1996)
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Long-term growth suppression of human glioma xenografts by chemoimmunoconjugates of 4-desacetylvinblastine-3-carboxyhydrazide and monoclonal antibody 9.2.27
Schrappe, M, Bumol, T F, Apelgren, L D, Briggs, S L, Koppel, G A, Markowitz, D D, Mueller, B M, Reisfeld, R A
Published in Cancer research (Chicago, Ill.) (15.07.1992)
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Published in Cancer research (Chicago, Ill.) (15.07.1992)
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Synthesis and structure-activity relationships of benzophenones as inhibitors of cathepsin D
Whitesitt, Celia A., Simon, Richard L., Reel, Jon K., Sigmund, Sandra K., Phillips, Michael L., Kevin Shadle, J., Heinz, Lawrence J., Koppel, Gary A., Hunden, David C., Lifer, Sherryl L., Berry, Dennis, Ray, Judy, Little, Sheila P, Xiadong Liu, Marshall, Winston S., Panetta, Jill A.
Published in Bioorganic & medicinal chemistry letters (17.09.1996)
Published in Bioorganic & medicinal chemistry letters (17.09.1996)
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A novel class of 5-HT2A receptor antagonists: aryl aminoguanidines
Bryant, H U, Nelson, D L, Button, D, Cole, H W, Baez, M B, Lucaites, V L, Wainscott, D B, Whitesitt, C, Reel, J, Simon, R, Koppel, G A
Published in Life sciences (1973) (01.09.1996)
Published in Life sciences (1973) (01.09.1996)
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Isolation of three separate anaphylatoxins from complement-activated human serum
Hugli, T E, Gerard, C, Kawahara, M, Scheetz, 2nd, M E, Barton, R, Briggs, S, Koppel, G, Russell, S
Published in Molecular and cellular biochemistry (01.12.1981)
Published in Molecular and cellular biochemistry (01.12.1981)
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A useful α, α′ - annulation reaction of enamines
Frontier, Alison J., Danishefsky, Samuel J., Koppel, Gary A., Meng, Dongfang
Published in Tetrahedron (15.10.1998)
Published in Tetrahedron (15.10.1998)
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BIOCHEMICAL AND MICROBIOLOGICAL STUDIES ON 7-METHOXYCEPHALOSPORINS
Ho, PETER P. K., TOWNER, RIDHARD D., INDELICATO, JOSEPH M., WILHAM, WILLIAM J., SPITZER, WAYNE A., KOPPEL, GARY A.
Published in Journal of antibiotics (01.01.1973)
Published in Journal of antibiotics (01.01.1973)
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Rapid parallel synthesis applied to the optimization of a series of potent nonpeptide neuropeptide Y-1 receptor antagonists
Siegel, Miles G., Chaney, Michael O., Bruns, Robert F., Clay, Michael P., Schober, Douglas A., Van Abbema, Anne M., Johnson, Douglas W., Cantrell, Buddy E., Hahn, Patric J., Hunden, David C., Gehlert, Donald R., Zarrinmayeh, Hamideh, Ornstein, Paul L., Zimmerman, Dennis M., Koppel, Gary A.
Published in Tetrahedron (24.09.1999)
Published in Tetrahedron (24.09.1999)
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A novel class of 5-HT 2a receptor antagonists: Aryl aminoguanidines
Bryant, Henry U., Nelson, David L., Button, Donald, Cole, Harlan W., Baez, Melvyn B., Lucaites, Virginia L., Wainscott, David B., Whitesitt, Cecilia, Reel, Jon, Simon, Richard, Koppel, Gary A.
Published in Life sciences (1973) (1996)
Published in Life sciences (1973) (1996)
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Synthetic Fc peptide-mediated regulation of the immune response. I: Characterization of the immunomodulating properties of a synthetic 23-amino acid peptide derived from the sequence of the CH3 domain of human IgG1
MORGAN, E. L, SHIELDS, J. E, CAMPBELL, C. S, BARTON, R. L, KOPPEL, G. A, WEIGLE, W. O
Published in The Journal of experimental medicine (01.03.1983)
Published in The Journal of experimental medicine (01.03.1983)
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Use of peptide combinatorial libraries in drug design: the identification of a potent serotonin reuptake inhibitor derived from a tripeptide cassette library
Koppel, Gary, Dodds, Carmen, Houchins, Brenda, Hunden, David, Johnson, Douglas, Owens, Rebecca, Chaney, Michael, Usdin, Theodore, Hoffman, Beth, Brownstein, Michael
Published in Chemistry & biology (01.07.1995)
Published in Chemistry & biology (01.07.1995)
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